DESIGN OF NEW ANTI-ALZHEIMER DRUGS: RING-EXPANSION SYNTHESIS AND SYNCHROTRON X-RAY DIFFRACTION STUDY OF DIMETHYL 4-ETHYL-11-FLUORO-1,4,5,6,7,8-HEXAHYDROAZONINO[5,6-B]INDOLE-2,3-DICARBOXYLATE СтатьяToze F.A.A., Listratova A.V., Voskressensky L.G., Chernikova N.Yu., Lobanov N.N., Bilyachenko A.N., Dorovatovskii P.V.Acta Crystallographica Section E: Crystallographic Communications. Том 74. 2018. С. 298-301
THREE-COMPONENT REACTION BETWEEN ISATOIC ANHYDRIDE, AMINE AND METH-YL-SUBS-TITUTED FURYL-ACRYL-ALDE-HYDES: CRYSTAL STRUCTURES OF 3-BENZYL-2-[(E)-2-(5-METHYLFURAN-2-YL)VIN-YL]-2,3-DI-HYDRO-QUINAZOLIN-4(1 H)-ONE, 3-BENZYL-2-[(E)-2-(FURAN-2-YL)-1-METHYL-VIN-YL]-2,3-DI-HYDRO-QUINAZOLIN-4(1 H)-ONE AND 3-(FURAN-2-YLMETH-YL)-2-[(E)-2-(FURAN-2-YL)-1-METHYL-VIN-YL]-2,3-DI-HYDRO-QUINAZOLIN-4(1 H)-ONE СтатьяZaytsev V.P., Sorokina E.A., Kvyatkovskaya E.A., Toze F.A.A., Mhaldar S.N., Dorovatovskii P.V., Khrustalev V.N.Acta Crystallographica Section E: Crystallographic Communications. Том 74. 2018. С. 1101-1106
CRYSTAL STRUCTURE OF 3-BENZYL-2-[(E)-2-(FURAN-2-YL)ETHENYL]-2,3-DIHYDROQUINAZOLIN-4(1H)-ONE AND 3-BENZYL-2-[(E)-2-(THIOPHEN-2-YL)ETHENYL]-2,3-DIHYDROQUINAZOLIN-4(1H)-ONE FROM SYNCHROTRON X-RAY DIFFRACTION СтатьяToze F.A.A., Zaytsev V.P., Chervyakova L.V., Kvyatkovskaya E.A., Dorovatovskii P.V., Khrustalev V.N.Acta Crystallographica Section E: Crystallographic Communications. Том 74. 2018. С. 10-14
CRYSTAL STRUCTURES OF (5RS)-(Z)-4-[5-(FURAN-2-YL)-3-PHENYL-4,5-DIHYDRO-1H-PYRAZOL-1-YL]-4-OXOBUT-2-ENOIC ACID AND (5RS)-(Z)-4-[5-(FURAN-2-YL)-3-(THIOPHEN-2-YL)-4,5-DIHYDRO-1H-PYRAZOL-1-YL]-4-OXOBUT-2-ENOIC ACID СтатьяBorisova K.K., Toze F.A.A., Yagafarov N.Z., Zubkov F.I., Dorovatovskii P.V., Zubavichus Y.V., Khrustalev V.N.Acta Crystallographica Section E: Crystallographic Communications. Том 72. 2016. С. 1557-1561
TRANSFORMATIONS OF 4-ARYLPYRROLO[1,2-A][1,4]BENZODIAZEPINES IN THREE-COMPONENT REACTIONS WITH ACTIVATED ALKYNES AND CH, NH, SH, AND OH ACIDS СтатьяVoskressensky L.G., Borisova T.N., Babakhanova M.I., Chervyakova T.M., Titov A.A., Novikov R.A., Toze F., Dang T.T.A., Varlamov A.V.Chemistry of Heterocyclic Compounds. Том 51. 2015. С. 639-646
TRANSFORMATIONS OF 4-ARYLPYRROLO[1,2-A][1,4]BENZODIAZEPINES IN THREE-COMPONENT REACTIONS WITH ACTIVATED ALKYNES AND СН, NH, SH, AND ОН ACIDS СтатьяVoskressensky L.G., Borisova T.N., Babakhanova M.I., Chervyakova T.M., Titov A.A., Novikov R.A., Toze F., Dang T.T.A., Varlamov A.V.Chemistry of Heterocyclic Compounds. Том Vol 51. 2015. С. 639-646
THE INTERACTION OF 4-HYDROXYMETHYL ISOINDOLINES WITH DEHYDROBENZENE. SYNTHESIS OF 3-PHENYLAMINOMETHYLDIHYDROBENZO[C]FURANES СтатьяVarlamov A.V., Guranova N.I., Borisova T.N., Toze F.A.A., Ovcharov M.V., Kristancho S., Voskressensky L.G.Tetrahedron. Том 71. 2015. С. 1175-1181
SYNTHESIS OF FURYL-, FURYLVINYL-, THIENYL-, PYRROLINYLQUINAZOLINES AND ISOINDOLO[2,1-A]QUINAZOLINES СтатьяZaytsev V.P., Revutskaya E.L., Kuźmenko M.G., Novikov R.A., Zubkov F.I., Sorokina E.A., Nikitina E.V., Toze F.A.A., Varlamov A.V.Russian Chemical Bulletin. Том 64. 2015. С. 1345-1353
CRYSTAL STRUCTURE OF METHYL (3RS,4SR,4ARS,11ARS,11BSR)-5-OXO-3,4,4A,5,7,8,9,10,11,11A-DECAHYDRO-3,11B-EPOXYAZEPINO[2,1-A]ISOINDOLE-4-CARBOXYLATE СтатьяToze F.A.A., Poplevin D.S., Zubkov F.I., Nikitina E.V., Porras C., Khrustalev V.N.Acta Crystallographica Section E: Crystallographic Communications. Том 71. 2015. С. o729-o730
SYNTHESIS OF 2-(CHLORO(METHOXY, MORPHOLINO)METHYL)-HEXAHYDROPYRIMIDOTHIENO[3,2-C]AZOCINES AND TETRAHYDROSPIRO[PYRIDO[4,5']THIENO[2,3-D]PYRIMIDINES] СтатьяVoskressensky L.G., Kovaleva S.A., Borisova T.N., Titov A.A., Toze F., Listratova A.V., Khrustalev V.N., Varlamov A.V.Chemistry of Heterocyclic Compounds. Том 51. 2015. С. 17-25
5-AMIDO- AND 5-AMINO-SUBSTITUTED EPOXYISOINDOLO[2,1-A]TETRAHYDROQUINOLINES AND 10-CARBOXYLIC ACIDS: THEIR SYNTHESIS AND REACTIVITY СтатьяZaytsev V.P., Zubkov F.I., Toze F.A.A., Orlova D.N., Eliseeva M.N., Grudinin D.G., Nikitina E.V., Varlamov A.V.Journal of Heterocyclic Chemistry. Том 50. 2013. С. E18-E38
RAC-METHYL (3AR*,4S*,5R*,7AR*)-5,7A-BIS(ACETYLOXY)- 3-OXO-2-PHENYLOCTAHYDRO-1H-ISOINDOLE-4-CARBOXYLATE СтатьяToze F.A.A., Nikitina E.V., Zaytsev V.P., Zubkov F.I., Khrustalev V.N.Acta Crystallographica Section E: Structure Reports Online. Том 69. 2013. o1555 с.
METHYL (9AR*,10S*,11R*,13AS*,13BS*)-9-OXO-6, 7,9,9A,10,11-HEXAHYDRO-5H,13BH-11,13A-EPOXYPYRROLO-[2′,1′:3,4][1,4] DIAZEPINO[2,1-A]ISOINDOLE-10-CARBOXYLATE СтатьяToze F.A.A., Airiyan I.K., Nikitina E.V., Sorokina E.A., Khrustalev V.N.Acta Crystallographica Section E: Structure Reports Online. Том 67. 2011. С. o2852-o2853
8A-METHYL-5,6,8,8A,9,10-HEXA-HYDRO-10,12A-EPOXY-ISOINDOLO[1,2-A] ISOQUINOLINIUM IODIDE СтатьяToze F.A.A., Ershova J.D., Obushak M.D., Zubkov F.I., Khrustalev V.N.Acta Crystallographica Section E: Structure Reports Online. Том 66. 2010. С. o1388-o1389
FIRST EXAMPLE OF DIELS-ALDER REACTION IN THE 2,3,4,4A-TETRAHYDROQUINOLINE SERIES. SYNTHESIS OF HYDROGENATED 5,8-ETHANOQUINOLINES СтатьяNikitina E.V., Khrustalev V.N., Grudinin D.G., Toze F.A.A., Kouznetsov V.V., Zubkov F.I.Tetrahedron. Том 66. 2010. С. 2889-2894