7th International Congress on Ultra Modern Telecommunications and Control Systems and Workshops, ICUMT 2015. Brno, Czech Republic, October 06-08, 2015.. Vol. 2016-January. 2016. P.. 243-246
Michael addition to unprotected 3-(2-nitrovinyl)indoles under the conditions of microwave synthesis
A novel highly efficient preparative method for the synthesis of substituted indoles using conjugate addition of nucleophiles to 3-(2-nitrovinyl)indoles has been developed. The addition of nucleophiles generated in the presence of a base from CH acids was investigated. The studied reactions proceed quickly and smoothly under the conditions of microwave activation and do not require protection of the indole nitrogen atom. © 2016 Springer Science+Business Media New York.
Authors
Aksenov A.V. 1 , Aksenov N.A. 1, 2 , Skomorokhov A.A. 1 , Aksenova I.V. 1 , Gryaznov G.D. 1 , Voskressensky L.G. 2 , Rubin M.A. 1, 3
Publisher
Латвийский институт органического синтеза Латвийской академии наук / Springer New York Consultants Bureau
Issue number
11
Language
English
Pages
923-927
State
Published
Link
Volume
52
Year
2016
Organizations
- 1 North-Caucasus Federal University, 1а Pushkin St., Stavropol, 355009, Russian Federation
- 2 Peoples’ Friendship University of Russia, 6 Miklukho-Maklaya St., Moscow, 117198, Russian Federation
- 3 The University of Kansas, 1251 Wescoe Hall Dr., Lawrence, KS 66045-7582, United States
Keywords
Addition; Indole; Michael reaction; Nitroalkenes
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Other records
Synthesis. Vol. 48. 2016. P.. 615-643